BDBM250499 US9464044, 141
SMILES NC(=O)C12CC3CC(C1)[C@H](NC(=O)C1(CNC(=O)N4CCCc5ccccc45)CC1)C(C3)C2
InChI Key InChIKey=BGURPVHOAXFRIQ-ZXSQAWDASA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 250499
Affinity DataIC50: 52.5nMpH: 6.0 T: 2°CAssay Description:The inhibiting activity of 11β-HSD1 derived from microsomal fractions was measured using the HTRF assay (62CO2PEB, Cisbio). Different concentrat...More data for this Ligand-Target Pair