BDBM260573 US10300066, Compound 47::US9532990, 47

SMILES COC(=O)NC(=O)\C=C/C(=O)N1CCCC(C1)n1nc(-c2ccc(Oc3c(F)c(F)cc(F)c3F)cc2F)c2c(N)ncnc12

InChI Key InChIKey=DTUMVLARIAWZBH-SREVYHEPSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 260573   

TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Zhejiang Dtrm Biopharma

US Patent
LigandPNGBDBM260573(US10300066, Compound 47 | US9532990, 47)
Affinity DataIC50:  6nMAssay Description:The enzyme reaction mixture of BTK wild type standard HTRF assay contained 1 nM BTK wild type, 1 μM biotin-TK1 peptide, and 30 μM ATP in a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Zhejiang Dtrm Biopharma

US Patent
LigandPNGBDBM260573(US10300066, Compound 47 | US9532990, 47)
Affinity DataIC50:  6nMT: 2°CAssay Description:The enzyme reaction mixture of BTK wild type standard HTRF assay contained 1 nM BTK wild type, 1 μM biotin-TK1 peptide, and 30 μM ATP in a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent