BDBM263546 2-{5-amino-1-[2-chloro-4-(3- cyano-phenoxy)-phenyl]-1h- pyrazole-4-carbonyl}-1h-indole- 5-carboxylic acid::US9556150, i-34
SMILES Nc1c(cnn1-c1ccc(Oc2cccc(c2)C#N)cc1Cl)C(=O)c1cc2cc(ccc2[nH]1)C(O)=O
InChI Key InChIKey=ULFBTRQJBNUGPM-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 263546
Affinity DataIC50: 25.1nMpH: 7.15Assay Description:This BTK competition assay measures compound potency (IC50) for the inactivated state of Bruton's Tyrosine Kinase using FRET (Förster/Fluorescenc...More data for this Ligand-Target Pair