BDBM263565 2-(4-{5-amino-4-[5-(3- dimethylamino-pyrrolidine-1- carbonyl)-1h-indole-2-carbonyl]- pyrazol-1yl}-3-chloro-phenoxy)- n,n-dimethyl-benzamide acetic acid salt::US9556150, i-53
SMILES CNC1CCN(C1)C(=O)c1ccc2[nH]c(cc2c1)C(=O)c1cnn(c1N)-c1ccc(Oc2ccccc2C(=O)N(C)C)cc1Cl
InChI Key
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 263565
Affinity DataIC50: 1.70nMpH: 7.15Assay Description:This BTK competition assay measures compound potency (IC50) for the inactivated state of Bruton's Tyrosine Kinase using FRET (Förster/Fluorescenc...More data for this Ligand-Target Pair