BDBM263966 2-(5-methyl-1H-pyrazol-1- yl)isonicotinic acid::US10173996, Example 31::US9604961, Example 31::US9714230, 31::US9908865, Example 31
SMILES Cc1ccnn1-c1cc(ccn1)C(O)=O
InChI Key InChIKey=DBNRSQHWQKIXGR-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 263966
Affinity DataIC50: 5.50E+3nMAssay Description:The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...More data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...More data for this Ligand-Target Pair