BDBM264041 2-[5-[(4-cyano-2- ethylphenyl)methoxy]pyrazol-1- yl]pyridine-4-carboxylic acid::US10173996, Example 126::US9604961, Example 126::US9714230, 126::US9908865, Example 126

SMILES CCc1cc(ccc1COc1ccnn1-c1cc(ccn1)C(O)=O)C#N

InChI Key InChIKey=LFHDOSKLOQHEPU-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 264041   

TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM264041(2-[5-[(4-cyano-2- ethylphenyl)methoxy]pyrazol-1- y...)
Affinity DataIC50: <100nMAssay Description:The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM264041(2-[5-[(4-cyano-2- ethylphenyl)methoxy]pyrazol-1- y...)
Affinity DataIC50:  550nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM264041(2-[5-[(4-cyano-2- ethylphenyl)methoxy]pyrazol-1- y...)
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent