BDBM264041 2-[5-[(4-cyano-2- ethylphenyl)methoxy]pyrazol-1- yl]pyridine-4-carboxylic acid::US10173996, Example 126::US9604961, Example 126::US9714230, 126::US9908865, Example 126
SMILES CCc1cc(ccc1COc1ccnn1-c1cc(ccn1)C(O)=O)C#N
InChI Key InChIKey=LFHDOSKLOQHEPU-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 264041
Affinity DataIC50: <100nMAssay Description:The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...More data for this Ligand-Target Pair
Affinity DataIC50: 550nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...More data for this Ligand-Target Pair