BDBM264081 5-(1-phenylethyl)-2-[4-(1H- tetrazol-5-yl)pyridin-2-yl]pyrazol- 3-ol::US10173996, Example 166::US9604961, Example 166::US9714230, 166::US9908865, Example 166

SMILES CC(c1cc(O)n(n1)-c1cc(ccn1)-c1nn[nH]n1)c1ccccc1

InChI Key InChIKey=NDZPISWATWIEPJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 264081   

TargetLysine-specific demethylase 2B(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM264081(5-(1-phenylethyl)-2-[4-(1H- tetrazol-5-yl)pyridin-...)
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM264081(5-(1-phenylethyl)-2-[4-(1H- tetrazol-5-yl)pyridin-...)
Affinity DataIC50:  5.50E+3nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent