BDBM264087 2-[3-[(3,5- dichlorophenyl)methyl]-5- hydroxypyrazol-1-yl]pyridine-4- carboxylic acid::US10173996, Example 172::US9604961, Example 172::US9714230, 172::US9908865, Example 172

SMILES OC(=O)c1ccnc(c1)-n1nc(Cc2cc(Cl)cc(Cl)c2)cc1O

InChI Key InChIKey=VNKGLVYANHHHFT-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 264087   

TargetLysine-specific demethylase 2B(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM264087(2-[3-[(3,5- dichlorophenyl)methyl]-5- hydroxypyraz...)
Affinity DataIC50:  550nMAssay Description:The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM264087(2-[3-[(3,5- dichlorophenyl)methyl]-5- hydroxypyraz...)
Affinity DataIC50:  5.50E+3nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent