BDBM268472 N-(6-cyclopropyl-7-(((trans)-4-(trifluoromethyl)cyclohexyl)-methoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)methanesulfonamide::US9550775, 13

SMILES CS(=O)(=O)Nc1nnc2cc(OC[C@H]3CC[C@@H](CC3)C(F)(F)F)c(cn12)C1CC1

InChI Key InChIKey=SNLBENSIDDPCRQ-AULYBMBSSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 268472   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM268472(N-(6-cyclopropyl-7-(((trans)-4-(trifluoromethyl)cy...)
Affinity DataIC50:  22.6nMpH: 7.2Assay Description:The following patch voltage clamp electrophysiology studies were performed on representative compounds of the invention using human embryonic kidney ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent