BDBM270924 4-(cyclohex-1-en-1-yl)-7-[(4-methylbenzene)sulfonyl]-5H-pyrrolo[3,2-d]pyrimidin-6-amine::US10059713, Example 42
SMILES Cc1ccc(cc1)S(=O)(=O)c1c(N)[nH]c2c(ncnc12)C1=CCCCC1
InChI Key InChIKey=NJEDVWCVFKBJMR-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 270924
Affinity DataEC50: 32nMAssay Description:GPR43 agonist/PAM activity was determined by measuring changes in intracellular calcium levels using a Ca2+ sensitive fluorescent dye. The changes in...More data for this Ligand-Target Pair