BDBM272154 (R)-5-(3-Fluoro-2-methylphenyl)-N-hydroxy-2-(5- fluoropyridin-2-yl)-5,6-dihydroxy-4H- cyclopenta[d]thiazole-5-carboxamide::US10065948, 96::US10457675, Example 96

SMILES Cc1c(F)cccc1[C@]1(Cc2nc(sc2C1)-c1ccc(F)cn1)C(=O)NO

InChI Key InChIKey=DTQZSNICTXHRFE-LJQANCHMSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 272154   

TargetHistone deacetylase 9(Homo sapiens (Human))
Chdi Foundation

US Patent
LigandPNGBDBM272154((R)-5-(3-Fluoro-2-methylphenyl)-N-hydroxy-2-(5- fl...)
Affinity DataIC50:  51nMAssay Description:The potency of the compounds is quantified by measuring the Histone Deacetylase 9 (HDAC9) enzymatic activity using the fluorogenic substrate, Boc-Lys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 9(Homo sapiens (Human))
Chdi Foundation

US Patent
LigandPNGBDBM272154((R)-5-(3-Fluoro-2-methylphenyl)-N-hydroxy-2-(5- fl...)
Affinity DataIC50:  51nMAssay Description:The potency of the compounds is quantified by measuring the Histone Deacetylase 9 (HDAC9) enzymatic activity using the fluorogenic substrate, Boc-Lys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent