BDBM275230 1-[(3S,4R)-1-methyl-4-(5- methylthiophen-2- yl)pyrrolidin-3-yl]-3-[1-(2- methylpyridin-4-yl)-1H- pyrazolo[3,4-c]pyridin-5- yl)urea::US9884048, Example 124::US9884048, Example 188
SMILES CN1C[C@@H](NC(=O)Nc2cc3cnn(-c4ccnc(C)c4)c3cn2)[C@@H](C1)c1ccc(C)s1
InChI Key InChIKey=APQXGNCZLGMYPP-RTBURBONSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 275230
Affinity DataIC50: 70nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair
Affinity DataIC50: 1.01nMAssay Description:Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each compound was dete...More data for this Ligand-Target Pair