BDBM275838 5-chloro-N-(N,N- dimethylsulfamoyl)-2- fluoro-4-(4-methoxy- phenethoxy)benzamide::US10071957, Example 57

SMILES COc1ccc(CCOc2cc(F)c(cc2Cl)C(=O)NS(=O)(=O)N(C)C)cc1

InChI Key InChIKey=SZVOFVWKETTWQX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 275838   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM275838(5-chloro-N-(N,N- dimethylsulfamoyl)-2- fluoro-4-(4...)
Affinity DataIC50:  2.40E+3nMpH: 7.4 T: 2°CAssay Description:Preparation of membranes containing recombinantly expressed sodium channels: Frozen recombinant cell pellets were thawed on ice and diluted to 4 time...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent