BDBM281291 US10022354, Example 231
SMILES [H][C@@]1(C[C@@H]1F)C(=O)N[C@@H]1CCN(C1)C(=O)c1cc(n[nH]1)C(C)C
InChI Key InChIKey=LXGAOGLHQMPZIY-VWYCJHECSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 281291
Affinity DataIC50: 0.330nMpH: 7.0 T: 2°CAssay Description:Full length KDM5A enzyme was expressed and purified inhouse. Biotin-H3K4me3 peptide was purchased from New England Biolabs. HTRF reagents (containing...More data for this Ligand-Target Pair