BDBM284977 N-(2-hydroxyethyl)-3-(2-methyl-1- oxoisoquinolin-4-yl)benzenesulfonamide::US10023592, Example 22
SMILES Cn1cc(-c2cccc(c2)S(=O)(=O)NCCO)c2ccccc2c1=O
InChI Key InChIKey=YBESZWZXEMEZKT-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 284977
Affinity DataIC50: 2.75E+3nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair