BDBM284980 4-(3-amino-5-fluorophenyl)-2- methylisoquinolin-1-one::US10023592, Example 25::US10941160, Example 25
SMILES Cn1cc(-c2cc(N)cc(F)c2)c2ccccc2c1=O
InChI Key InChIKey=HFXJXEJLKHMMSN-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 284980
Affinity DataIC50: 2.75E+3nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: 2.75E+3nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair