BDBM285098 4-[5-(cyclopropylmethoxy)-2- (methylsulfonylmethyl)pyrimidin-4-yl]-2- methylisoquinolin-1-one::US10023592, Example 143
SMILES Cn1cc(-c2nc(CS(C)(=O)=O)ncc2OCC2CC2)c2ccccc2c1=O
InChI Key InChIKey=YVEZTYYLJSOPFM-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 285098
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair