BDBM285296 2-methyl-4-(3-methylsulfonyl-5- phenylmethoxyphenyl)isoquinolin-1-one::BDBM486140::US10023592, Example 344
SMILES Cn1cc(-c2cc(OCc3ccccc3)cc(c2)S(C)(=O)=O)c2ccccc2c1=O
InChI Key InChIKey=FKWDUYPFNXYDTJ-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 285296
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair
Affinity DataIC50: <500nMpH: 7.3Assay Description:Determination of the IC50 for the heterocyclic derivative BRD4 inhibitors disclosed herein was performed as follows. His-tagged BRD4 was cloned, expr...More data for this Ligand-Target Pair