BDBM289081 US10093650, Example 24::US11479538, Example 24

SMILES CCc1ccc(s1)C1=C(C(=O)N[C@@H](C1)c1ccc(OCCCC(F)(F)F)cc1Cl)n1nn[nH]c1=O

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 289081   

Target2-acylglycerol O-acyltransferase 2(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM289081(US10093650, Example 24 | US11479538, Example 24)
Affinity DataIC50:  36nMAssay Description:The MGAT enzyme reactions were performed in Corning FALCONŽ 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAlpha-1,6-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase(Homo sapiens (Human))
Bristol-Myers Squibb

US Patent
LigandPNGBDBM289081(US10093650, Example 24 | US11479538, Example 24)
Affinity DataIC50:  36nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCONŽ 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent