BDBM289446 5-(2-cyclopropyl-1-(3-(oxazol-5-yl)bicyclo[1.1.1]pentan-1-yl)-1H-imidazol-4-yl)-3-(trifluoromethoxy)pyridin-2-amine::US10093664, Example 27

SMILES Nc1ncc(cc1OC(F)(F)F)-c1cn(c(n1)C1CC1)C12CC(C1)(C2)c1cnco1

InChI Key InChIKey=DOTWXGYHTFWCEU-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 289446   

TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289446(5-(2-cyclopropyl-1-(3-(oxazol-5-yl)bicyclo[1.1.1]p...)
Affinity DataKd:  29nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent