BDBM289449 5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-(tetrahydrofuran- 3-yl)-1H-imidazol-4- yl)-3-(trifluoro- methoxy)pyridin-2- amine::US10093664, Example 30

SMILES Nc1ncc(cc1OC(F)(F)F)-c1cn(c(n1)C1CCOC1)C12CC(C1)(C2)N1CCOCC1

InChI Key InChIKey=ZBFPMRVKWIXRQL-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 289449   

TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289449(5-(1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-2-...)
Affinity DataKd:  390nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent