BDBM289505 1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-1-(3-morpholino- bicyclo[1.1.1]pentan-1- yl)-1H-imidazol-2-yl)- 2,2,2-trifluoroethan-1- ol::US10093664, Example 69a

SMILES Nc1ncc(cc1C(F)(F)F)-c1cn(c(n1)C(O)C(F)(F)F)C12CC(C1)(C2)N1CCOCC1

InChI Key InChIKey=YZHZXQQOTGYMHG-UHFFFAOYSA-N

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 289505   

TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM289505(1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-...)
Affinity DataKd:  0.360nMAssay Description:The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent