BDBM294008 (2S)-5-(1-(1H-Tetrazol-5- yl)pent-3-yn-2-yl)-2-((3-(2- methylphenyl)benzo[b]thiophen- 5-yl)methoxy)pyridine::US10106553, Compound 40

SMILES CC#C[C@@H](Cc1nnn[nH]1)c1ccc(OCc2ccc3scc(-c4ccccc4C)c3c2)nc1

InChI Key

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 294008   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM294008((2S)-5-(1-(1H-Tetrazol-5- yl)pent-3-yn-2-yl)-2-((3...)
Affinity DataEC50:  58nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent