BDBM294385 US9586959, Compound 48
SMILES CNC1CN(C1)c1nc2ncc(I)cc2n2cnnc12
InChI Key InChIKey=SGQVHLLHCYFWEE-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 294385
Affinity DataIC50: 65nMpH: 7.5 T: 2°CAssay Description:In vitro profiling protein kinases was performed using the HotSpot assay platform. Briefly, specific kinase/substrate pairs along with required cofac...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+7nMAssay Description:The binding assays of the human serotonin 3 receptor for present invention were performed at Cerep (Poitiers, France).More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+8nMpH: 7.4 T: 2°CAssay Description:Each compound of the present invention prepared in the examples was prepared in DMSO into concentrations of 0.02, 0.06, 0.3 and 2 mM. 10 uL of the pr...More data for this Ligand-Target Pair