BDBM299143 (6R,8R)-6-(4-(2- (3- (fluoromethyl) azetidin-1- yl)ethoxy) phenyl)-7-((3- fluorooxetan-3- yl)methyl)-6,8- dimethyl-6,7,8,9- tetrahydro-3H- pyrazolo[4,3- f]isoquinoline::US10125135, Example 32
SMILES C[C@@H]1Cc2c(ccc3[nH]ncc23)[C@](C)(N1CC1(F)COC1)c1ccc(OCCN2CC(CF)C2)cc1
InChI Key
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 299143
Affinity DataIC50: 0.670nMAssay Description:The ability of compounds to bind to isolated Estrogen Receptor Alpha Ligand binding domain (ER alpha LBD (GST)) was assessed in competition assays us...More data for this Ligand-Target Pair