BDBM306780 N1-(5- ((1R,3R)-2-((3- fluorooxetan- 3-yl)methyl)- 3-methyl- 2,3,4,9- tetrahydro-1H- pyrido[3,4- b]indol-1-yl)- 4-methoxy- pyridin-2- yl)-N2-(3- fluoropropyl) ethane-1,2- diamine::US10149839, Example 66
SMILES COc1cc(NCCNCCCF)ncc1[C@H]1N(CC2(F)COC2)[C@H](C)Cc2c1[nH]c1ccccc21
InChI Key
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 306780
Affinity DataIC50: 1nMAssay Description:The ability of compounds to down-regulate Estrogen Receptor (ER) numbers was assessed in a cell based immuno-fluorescence assay using the MCF-7 human...More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Compounds were dosed directly from a compound source microplate containing serially diluted compound (4 wells containing 10 mM, 0.1 mM, 1 mM and 10 n...More data for this Ligand-Target Pair