BDBM309344 N-(6-(4-(4-fluorophenoxy)phenyl)pyridin-2-yl)cyclopropaneSulfonamide::US9656959, Example 28

SMILES Fc1ccc(Oc2ccc(cc2)-c2cccc(NS(=O)(=O)C3CC3)n2)cc1

InChI Key InChIKey=CAJGZYDAWGNVNQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 309344   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Purdue Pharma

US Patent
LigandPNGBDBM309344(N-(6-(4-(4-fluorophenoxy)phenyl)pyridin-2-yl)cyclo...)
Affinity DataIC50:  220nMAssay Description:In vitro assays were performed in a recombinant cell line expressing cDNA encoding the alpha subunit (Nav1.7, SCN9a, PN1, NE) of human Nav1.7 (Access...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent