BDBM309910 1- (benzo[c][1,2,5]thia- diazol-5-yl)-3-(1H- benzo[d]imidazol-5- yl)thiourea::US9656991, 24

SMILES S=C(Nc1ccc2[nH]cnc2c1)Nc1ccc2nsnc2c1

InChI Key InChIKey=OUIZUDZKLFGCEN-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 309910   

TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

US Patent
LigandPNGBDBM309910(1- (benzo[c][1,2,5]thia- diazol-5-yl)-3-(1H- benzo...)
Affinity DataKi:  4.93E+3nMAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

US Patent
LigandPNGBDBM309910(1- (benzo[c][1,2,5]thia- diazol-5-yl)-3-(1H- benzo...)
Affinity DataIC50:  3.24E+4nMAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrates. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent