BDBM311520 5-{[cis-2- aminocyclohexyl]amino}- N-(3-carbamoyl-1- pyridin-3-yl-1H- pyrazol-4- yl)pyrazolo[1,5- a]pyrimidine-3- carboxamide::US10155765, Example 6
SMILES N[C@@H]1CCCC[C@@H]1Nc1ccn2ncc(C(=O)Nc3cn(nc3C(N)=O)-c3cccnc3)c2n1
InChI Key InChIKey=TYFNEYCNSDXOTM-CVEARBPZSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 311520
Affinity DataIC50: 0.800nMAssay Description:The kinase activity of IRAK4 is determined by its ability to catalyze the phosphorylation of a fluorescent polypeptide substrate. The extent of phosp...More data for this Ligand-Target Pair