BDBM318664 (4S)-7-(3,5-dimethylisoxazol-4-yl)-2- [(8aS)-hexahydropyrrolo[1,2-a]pyrazin- 2(1H)-yl]-4-pyridin-2-yl-4,5- dihydroimidazo[1,5,4- de][1,4]benzoxazine::US10464947, Example 193A::US9624241, Example 193A
SMILES Cc1noc(C)c1-c1ccc2nc(N3CCN4CCC[C@H]4C3)n3[C@H](COc1c23)c1ccccn1
InChI Key InChIKey=WKAPWJJIVIHBPA-PGRDOPGGSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 318664
Affinity DataIC50: <100nMAssay Description:BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for BD2. Inhib...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 40 μL for BD1 and 60 μL for BD2. Inhib...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:BRD4-BD1 and BRD4-BD2 assays were conducted in white 384-well polystyrene plate in a final volume of 20 μL for BD1 and 40 μL for BD2. Inhib...More data for this Ligand-Target Pair