BDBM319678 2-[5-(4-fluorophenyl)-1-methyl-1H-imidazol-4-yl]-4- [5-(trifluoromethyl)-1H-1,2,3-triazol-4-yl]pyridine::US10174003, Example 97::US9896436, Example 97

SMILES Cn1cnc(c1-c1ccc(F)cc1)-c1cc(ccn1)-c1nn[nH]c1C(F)(F)F

InChI Key InChIKey=KDDMSZINJMDMMC-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 319678   

TargetLysine-specific demethylase 2B(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM319678(2-[5-(4-fluorophenyl)-1-methyl-1H-imidazol-4-yl]-4...)
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of FBXL10 was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 6B(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM319678(2-[5-(4-fluorophenyl)-1-methyl-1H-imidazol-4-yl]-4...)
Affinity DataIC50: >1.00E+4nMAssay Description:The ability of test compounds to inhibit the activity of JMJD3 was determined in 384-well plate format under the following reaction conditions: 1 nM ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM319678(2-[5-(4-fluorophenyl)-1-methyl-1H-imidazol-4-yl]-4...)
Affinity DataIC50: >1.00E+4nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM319678(2-[5-(4-fluorophenyl)-1-methyl-1H-imidazol-4-yl]-4...)
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent