BDBM320310 2-({3,7-Bis[4-(2H3)methyl-1-methyl-1H-1,2,3-triazol-5-yl]-5H-pyrido[3,2-b]indol-5-yl}(oxan-4-yl)methyl)-3-fluoropyridine::US10174024, Example 27::US10174024, Example 28
SMILES Cc1nnn(C)c1-c1ccc2c(c1)n(C(C1CCOCC1)c1ncccc1F)c1cc(cnc21)-c1c(C)[nH]nn1C
InChI Key InChIKey=ZXBNXJZSTOXWGH-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 320310
Affinity DataIC50: <5nMAssay Description:The binding of compounds to bromodomain BRD4 (44-168), BRD4 (333-460), and BRD4 (1-477 or 44-460) was assessed using a time resolved fluorescent reso...More data for this Ligand-Target Pair
Affinity DataIC50: <5nMAssay Description:The binding of compounds to bromodomain BRD4 (44-168), BRD4 (333-460), and BRD4 (1-477 or 44-460) was assessed using a time resolved fluorescent reso...More data for this Ligand-Target Pair