BDBM320379 2-[hydroxy-(3-methyl- phenyl)methyl]-1H-pyrrolo[3,2- b]pyridine-7-carboxylic acid::US10174026, Example 22::US9738637, Example 22

SMILES Cc1cccc(c1)C(O)c1cc2nccc(C(O)=O)c2[nH]1

InChI Key

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 320379   

TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Celgene Quantical Research

US Patent
LigandPNGBDBM320379(2-[hydroxy-(3-methyl- phenyl)methyl]-1H-pyrrolo[3,...)
Affinity DataIC50: <100nMAssay Description:The enzymatic assay of Jarid1A activity is based upon Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The ability of test c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 4C(Homo sapiens (Human))
Celgene Quantical Research

US Patent
LigandPNGBDBM320379(2-[hydroxy-(3-methyl- phenyl)methyl]-1H-pyrrolo[3,...)
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Celgene Quantical Research

US Patent
LigandPNGBDBM320379(2-[hydroxy-(3-methyl- phenyl)methyl]-1H-pyrrolo[3,...)
Affinity DataIC50: <100nMAssay Description:The ability of test compounds to inhibit the activity of Jarid1B was determined in 384-well plate format under the following reaction conditions: 0.8...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent