BDBM323175 N-[(S)-1-[(S)-2-(3-hydroxy-3-o-tolylazetidin-1-yl)-1-(4-methoxybenzyl)-2-oxoethylcarbamoyl]-2-(1H-imidazol-4-yl)ethyl]benzamide::US9630949, 4

SMILES COc1ccc(C[C@H](NC(=O)[C@H](Cc2c[nH]cn2)NC(=O)c2ccccc2)C(=O)N2CC(O)(C2)c2ccccc2C)cc1

InChI Key InChIKey=LGFFOUNKABARGH-VMPREFPWSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 323175   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM323175(N-[(S)-1-[(S)-2-(3-hydroxy-3-o-tolylazetidin-1-yl)...)
Affinity DataEC50:  4.00E+3nMAssay Description:In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Galderma Research & Development

US Patent
LigandPNGBDBM323175(N-[(S)-1-[(S)-2-(3-hydroxy-3-o-tolylazetidin-1-yl)...)
Affinity DataEC50:  250nMAssay Description:In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent