BDBM323616 (E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl)phenoxy)hex-2-enoic acid ::US10188627, Compound 8cc

SMILES CN(Cc1ccccc1OCCC\C=C\C(O)=O)C(=O)c1ccc(cc1)-c1ccco1

InChI Key InChIKey=PRLUQZAEJIZRCO-QDEBKDIKSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 323616   

TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Mitobridge

US Patent
LigandPNGBDBM323616((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Affinity DataEC50:  80.4nMAssay Description:Medium including test compound was aspirated and washed with PBS. 50 μl PBS including 1 mM Mg++ and Ca++ were then added to each well. The lucif...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Mitobridge

Curated by ChEMBL
LigandPNGBDBM323616((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human PPARgamma LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Mitobridge

Curated by ChEMBL
LigandPNGBDBM323616((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human PPARalpha LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Mitobridge

US Patent
LigandPNGBDBM323616((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Affinity DataEC50:  80nMAssay Description:Activation of human PPARdelta LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed