BDBM3255 4-Anilino quinazoline deriv. 6::N-(2-phenylethyl)quinazolin-4-amine

SMILES C(Cc1ccccc1)Nc1ncnc2ccccc12

InChI Key InChIKey=YKOSADJQCBRMRR-UHFFFAOYSA-N

Data  1 KI  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 3255   

TargetAdenosine receptor A2a(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM3255(4-Anilino quinazoline deriv. 6 | N-(2-phenylethyl)...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane incubated for 1 hr by microplate beta scintillation ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Human)
University of Auckland

LigandPNGBDBM3255(4-Anilino quinazoline deriv. 6 | N-(2-phenylethyl)...)
Affinity DataIC50:  4.10E+3nMpH: 7.4 T: 22°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed