BDBM327965 5-(4-(4- fluorobenzyl)piperazine- 1-carbonyl)-N-(cis-3- fluoropiperidin-4- yl)picolinamide::US10377742, Compound 102::US9663496, Compound 102

SMILES F[C@H]1CNCC[C@H]1NC(=O)c1ccc(cn1)C(=O)N1CCN(Cc2ccc(F)cc2)CC1

InChI Key InChIKey=SSXKELDQHCLBAC-VQTJNVASSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 327965   

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Homo sapiens (Human))
Rigel Pharmaceuticals

US Patent
LigandPNGBDBM327965(5-(4-(4- fluorobenzyl)piperazine- 1-carbonyl)-N-(c...)
Affinity DataEC50:  7.50E+3nMAssay Description:Compounds were assayed for their ability to activate AMPK using an enzyme-linked immunosorbent assay. Reagents and procedures for measuring AMPK acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Homo sapiens (Human))
Rigel Pharmaceuticals

US Patent
LigandPNGBDBM327965(5-(4-(4- fluorobenzyl)piperazine- 1-carbonyl)-N-(c...)
Affinity DataEC50:  7.50E+3nMAssay Description:Compounds were assayed for their ability to activate AMPK using an enzyme-linked immunosorbent assay. Reagents and procedures for measuring AMPK acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent