BDBM329232 4-(5-chloro-6-((trans-3-methylcyclobutyl)oxy)-3-pyridinyl)-2-::4-(5-chloro-6-((trans-3-methylcyclobutyl)oxy)-3-pyridinyl)-2-fluoro-5-methoxy-N-(methylsulfonyl)benzamide::US9663508, Example 735

SMILES COc1cc(C(=O)NS(C)(=O)=O)c(F)cc1-c1cnc(O[C@H]2C[C@H](C)C2)c(Cl)c1

InChI Key InChIKey=NKZOJBBRMNWKSB-UMSPYCQHSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 329232   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM329232(4-(5-chloro-6-((trans-3-methylcyclobutyl)oxy)-3-py...)
Affinity DataIC50:  59.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent