BDBM329301 4-(5-chloro-6-(cyclobutyloxy)- 3-pyridinyl)-5-cyclopropyl-2- fluoro-N- (methylsulfonyl)benzamide::4-(5-chloro-6-(cyclobutyloxy)-3-pyridinyl)-5-cyclopropyl-2-fluoro-N-(methylsulfonyl)benzamide::US9663508, Example 802

SMILES CS(=O)(=O)NC(=O)c1cc(C2CC2)c(cc1F)-c1cnc(OC2CCC2)c(Cl)c1

InChI Key InChIKey=WDTVVGOSLYOENZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 329301   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM329301(4-(5-chloro-6-(cyclobutyloxy)- 3-pyridinyl)-5-cycl...)
Affinity DataIC50:  136nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent