BDBM329768 Preparation of 2-[6-(4-chlorophenyl)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1]benzazepin-4-yl]-1-(8-oxa-3-azabicyclo[3.2.1]oct-3-yl)ethanone::US9663523, Example 32
SMILES Cc1nnc2C(CC(=O)N3CC4CCC(C3)O4)C=C(c3ccc(Cl)cc3)c3ccccc3-n12
InChI Key InChIKey=CWFCPLBUIOLJBW-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 329768
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Bayer Pharma Aktiengesellschaft
US Patent
Bayer Pharma Aktiengesellschaft
US Patent
Affinity DataIC50: 390nMAssay Description:For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...More data for this Ligand-Target Pair