BDBM330426 4-{S-methyl-N-[(5-{4-[4-({[(3- methylphenyl)amino]carbonyl} amino)phenoxy]pyridin-2-yl}- 1H-pyrrol-3-yl)carbonyl] sulfonimidoyl}butanoic acid::US9725433, 82

SMILES Cc1cccc(NC(=O)Nc2ccc(Oc3ccnc(c3)-c3cc(c[nH]3)C(=O)N=S(C)(=O)CCCC(O)=O)cc2)c1

InChI Key

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 330426   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Allergan

US Patent
LigandPNGBDBM330426(4-{S-methyl-N-[(5-{4-[4-({[(3- methylphenyl)amino]...)
Affinity DataIC50:  19nMAssay Description:Automated FLIPR (Fluorometric Imaging Plate Reader) technology was used to screen for inhibitors of VEGF induced increases in intracellular calcium l...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent