BDBM332504 4-[1-{[2-chloro-6- (trifluoromethyl) phenyl]carbonyl}-6- (1-methyl-1H-pyrazol- 5-yl)-1H-indazol- 3-yl]benzoic acid::US10196354, Example 23J::US9745265, 23J
SMILES Cn1nccc1-c1ccc2c(nn(C(=O)c3c(Cl)cccc3C(F)(F)F)c2c1)-c1ccc(cc1)C(O)=O
InChI Key InChIKey=BPUYMKDBEOEQSL-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 332504
Affinity DataIC50: >1.00E+4nMAssay Description:To identify novel antagonists of RORgammaT, an assay was developed which employs the interaction of RORgammaT with its co-activator peptide SRC1_2. T...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:The compounds of the invention inhibit RORgammaT activity. Activation of RORgammaT activity can be measured using, e.g., biochemical TR-FRET assay. I...More data for this Ligand-Target Pair