BDBM34149 CHEMBL94422::N-benzenesulfonylgramine antagonist, 8
SMILES CN(C)Cc1cn(c2ccccc12)S(=O)(=O)c1ccccc1
InChI Key InChIKey=MHFSWNYVTLJUEH-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 34149
Affinity DataKi: 3nM ΔG°: -12.1kcal/mole EC50: 880nMpH: 7.4 T: 37°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Antagonistic activity towards 5-hydroxytryptamine 6 receptor was evaluated in cAMP assayMore data for this Ligand-Target Pair