BDBM343296 N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-4-(6-methoxy-5-methylpyrimidin-4-yl)-1-methyl-1H-pyrazole-5-carboxamide::US9777000, Example 3.31

SMILES COc1ncnc(-c2cnn(C)c2C(=O)Nc2cc3nc(nn3cc2F)-c2ccccc2)c1C

InChI Key InChIKey=HNKMWNJVVZKLRX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 343296   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Mochida Pharmaceutical

US Patent
LigandPNGBDBM343296(N-(6-fluoro-2-phenyl-[1,2,4]triazolo[1,5-a]pyridin...)
Affinity DataIC50: <5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent