BDBM343399 4-(4,5-dimethylthiazol-2-yl)-1-methyl-N-(2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-1H-pyrazole-5-carboxamide::US9777000, Example 5.45

SMILES Cc1nc(sc1C)-c1cnn(C)c1C(=O)NC1CCn2nc(nc2C1)N1CCCC1

InChI Key InChIKey=OIBKAYBSCYCHLS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 343399   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Homo sapiens (Human))
Mochida Pharmaceutical

US Patent
LigandPNGBDBM343399(4-(4,5-dimethylthiazol-2-yl)-1-methyl-N-(2-(pyrrol...)
Affinity DataIC50: <5nMAssay Description:IMAP TR-FRET Phosphodiersterase Evaluation Assay Kit (Molecular Device) was used for the measurement. Ten μL of a diluted test compound having e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent