BDBM344936 1-[(4,5-dimethyl-1,3-::1-[(4,5-dimethyl-1,3-oxazol-2-yl)methyl]-3-[1-(2-fluorophenyl)-1H-indazol-4-yl]imidazolidin-2-one::US9783527, Example 238

SMILES Cc1nc(CN2CCN(C2=O)c2cccc3n(ncc23)-c2ccccc2F)oc1C

InChI Key InChIKey=GPLRUGBFKFEETM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 344936   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM344936(1-[(4,5-dimethyl-1,3- | 1-[(4,5-dimethyl-1,3-oxazo...)
Affinity DataIC50:  586nMAssay Description:Two days prior to the experiment, frozen HEK293 cells stably expressing recombinant human Nav1.7 were quickly thawed and plated at 25,000 cells/well ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent