BDBM345531 N-(6-(1,5-dimethyl-6-oxo-1,6- dihydropyridin-3-yl)-2-((1-methyl- 1H-indol-4-yl)oxy)pyrimidin-4- yl)propane-2-sulfonamide::US10202360, Example 76
SMILES CC(C)S(=O)(=O)Nc1cc(nc(Oc2cccc3n(C)ccc23)n1)-c1cc(C)c(=O)n(C)c1
InChI Key InChIKey=ADPWZHAESCQHBK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 345531
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the CREBBP inhibitors disclosed herein was performed as follows: CREBBP was cloned and expressed in E. Coli as His-tag ...More data for this Ligand-Target Pair