BDBM345582 Propane-2-sulfonic acid [6-(1,5- dimethyl-6-oxo-1,6-dihydro-pyridin- 3-yl)-2-(1-ethyl-3,5-dimethyl-1H- pyrazol-4-yloxy)-pyrimidin-4-yl]- amide::US10202360, Example 127
SMILES CCn1nc(C)c(Oc2nc(NS(=O)(=O)C(C)C)cc(n2)-c2cc(C)c(=O)n(C)c2)c1C
InChI Key InChIKey=XYDOXJAGTMVSMF-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 345582
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the CREBBP inhibitors disclosed herein was performed as follows: CREBBP was cloned and expressed in E. Coli as His-tag ...More data for this Ligand-Target Pair