BDBM345604 N-(2-(2-cyano-6-methylphenoxy)-6- (1-methyl-6-oxo-1,6- dihydropyridin-3-yl)pyrimidin-4-yl)- 3,3,3-trifluoropropane-1- sulfonamide::US10202360, Example 149

SMILES Cc1cccc(C#N)c1Oc1nc(NS(=O)(=O)CCC(F)(F)F)cc(n1)-c1ccc(=O)n(C)c1

InChI Key InChIKey=BELJQQRHBGKATE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 345604   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM345604(N-(2-(2-cyano-6-methylphenoxy)-6- (1-methyl-6-oxo-...)
Affinity DataIC50: <500nMAssay Description:Determination of the IC50 for the CREBBP inhibitors disclosed herein was performed as follows: CREBBP was cloned and expressed in E. Coli as His-tag ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent