BDBM346507 US10202378, Example 111::[2-(hydroxymethyl)phenyl]methyl4-(3-hydroxy-3-methyl-but-1-ynyl)-2,6-dimethyl-7-oxo-1H-pyrrolo[2,3-c]pyridine-3-carboxylate
SMILES Cc1[nH]c2c(c1C(=O)OCc1ccccc1CO)c(cn(C)c2=O)C#CC(C)(C)O
InChI Key InChIKey=XOLLFMCFALREEU-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 346507
TargetTranscription initiation factor TFIID subunit 1 [1381-1497](Homo sapiens (human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 259nMAssay Description:His/Flag epitope tagged TAF1-BD11381-1497 was cloned, expressed, and purified to homogeneity. TAF1-BD binding and inhibition was assessed by monitori...More data for this Ligand-Target Pair
TargetTranscription initiation factor TFIID subunit 1 [1504-1635](Homo sapiens (Human))
Genentech
US Patent
Genentech
US Patent
Affinity DataIC50: 37.9nMAssay Description:His/Flag epitope tagged TAF1-BD21504-1635 was cloned, expressed, and purified to homogeneity. TAF1-BD2 binding and inhibition was assessed by monitor...More data for this Ligand-Target Pair